Cyclobenzaprine

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Cyclobenzaprine
Identifiers
Brand Names: Apo-Cyclobenzaprine, Flexeril, Fexmid, Amrix
Slang Names: "Cyclone," "Mellow Yellow"
Chemical/Physical Properties
Solubility: Soluble in cold water.
Legal Status
US: UNSCHEDULED
Routes of Administration
Oral: Yes
Insufflation: No
Smoking: No
Intravenous: Yes, though uncommon
Intramuscular: Yes, though uncommon
Sublingual: Yes
Rectal: Yes

Cyclobenzaprine is a muscle relaxant that is active in the Central Nervous System and interacts with the signals sent to the muscles that cause them to tighten. It is often given to patients who suffer from pain and muscle spasms resulting from whiplash type injuries, and is effective at treating symptoms of fibromyalgia. It also works wonders at knocking you unconscious when enough is taken, otherwise it is a mild sedative.

Cyclobenzaprine is marketed as:

  • Apo-Cyclobenzaprine (10 mg tablets)
  • Flexeril (5 and 10 mg tablets) (Available as generic)
  • Fexmid (7.5 mg tablet) (Available as generic)
  • Amrix as a once a day ER (15 or 30 mg capsules)


Contents

[edit] Dosage

Doses are for those without tolerance. Remember, a recreational dose will vary from person to person depending on a variety of factors, such as build and interactions with other legal or illegal substances, including prescription medications. Best to check Google first. If you are mixing prescription medications. Check out this website: http://www.drugs.com/drug_interactions.php . Some of their interactions that they mention are a little too much or they are being cautious but its a good utility to have in case you ever need to check.

Cyclobenzaprine should NOT be taken along with any MAOI (monoamine oxidase inhibitor), as it could result in fatality.

Taken sublingually, cyclobenzaprine is noticeable within a few minutes, and is most often the preferred ROA. Take note, however, that dissolved cyclobenzaprine WILL make your mouth and tongue NUMB. This effect lasts for upwards of an hour, and isn't usually a problem unless you're retarded and bite your tongue a lot.

Low 5mg-15mg
Medium 15mg-30mg
High 30mg+

[edit] Common side effects

Effects and side effects are shared by most CNS depressants:

Short term

  • Sedation
  • Dizziness
  • Drymouth

Overdose

  • Convulsions
  • Ataxia
  • Tachycardia
  • Cardiac arrhythmia

[edit] As A Potentiator

Cyclobenzaprine steepens the dose-to-response curve of codeine and if taken with on an empty stomach can give the user a rush of euphoria[1]

[edit] References

Muscle Relaxant

Carisoprodol (Soma)

[edit] Links

MSDS[2]

DrugBank Page[3]

Wikipedia[4]

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